SCHEMBL8553071

SCHEMBL8553071

CCC(CC)N1CCC(c2csc3ccc(NC(=O)c4ccco4)cc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.47
MEN1 O00255 8/20 0.47
MAPT P10636 8/20 0.47
LMNA P02545 4/20 0.47
NPC1 O15118 11/20 0.43
RAB9A P51151 11/20 0.43
SMN1; SMN2 Q16637 8/20 0.42
HSD17B10 Q99714 4/20 0.42
TSHR P16473 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HPGD P15428 2/20 0.42
TP53 P04637 5/20 0.42
MAPK1 P28482 2/20 0.42
PKM P14618 2/20 0.42
GAA P10253 1/20 0.41
ALDH1A1 P00352 3/20 0.41
CASP1 P29466 2/20 0.41
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552316 0.88 NPC1 (0.54) KMT2AMEN1MAPTLMNANPC1
SCHEMBL8553073 0.84 DRD2 (0.46) KMT2AMEN1MAPTLMNANPC1
SCHEMBL8553184 0.84 RAB9A (0.41) NPC1RAB9ASMN1; SMN2TP53
SCHEMBL8548010 0.84 DRD2 (0.40) KMT2AMEN1MAPTKDM4EHPGD
SCHEMBL8549937 0.84 DRD2 (0.46) KMT2AMEN1MAPTLMNANPC1
SCHEMBL8704365 0.83 DRD2 (0.42) KMT2AMEN1MAPTLMNANPC1
SCHEMBL7476220 0.82 HTR1D (0.54)
SCHEMBL8552293 0.82 LMNA (0.42) KMT2AMEN1MAPTLMNAHSD17B10
SCHEMBL8723743 0.80 MAPT (0.47) KMT2AMEN1MAPTLMNANPC1
SCHEMBL8547967 0.78 MAPT (0.46) KMT2AMEN1MAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
WO-1998015545-A1 NEW SEROTONIN 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 1998-04-16 WO disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed