SCHEMBL8553525

SCHEMBL8553525

CCC=CCCOC(=O)Nc1ccc2scc(C3CCN(CCCCC)CC3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.43
SLC6A4 P31645 1/20 0.43
HTR1D P28221 10/20 0.37
HTR1B P28222 8/20 0.37
CHRM2 P08172 1/20 0.37
NPC1 O15118 4/20 0.37
RAB9A P51151 4/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
HPGD P15428 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
MAPT P10636 2/20 0.36
TP53 P04637 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
KMT2A Q03164 1/20 0.36
RELA Q04206 1/20 0.36
BCHE P06276 4/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553059 0.88 DRD2 (0.42) DRD2SLC6A4HTR1DHTR1BCHRM2
SCHEMBL8552203 0.87 CCR2 (0.43) DRD2SLC6A4HTR1DHTR1BCHRM2
SCHEMBL8553522 0.86 DRD2 (0.35) DRD2SLC6A4HTR1DHTR1BNPC1
SCHEMBL8549865 0.84 DRD2 (0.44) DRD2SLC6A4NPC1RAB9ASMN1; SMN2
SCHEMBL7481590 0.84 HTR1D (0.56) DRD2HTR1DHTR1BCHRM2
SCHEMBL8552297 0.81 DRD2 (0.48) DRD2SLC6A4
SCHEMBL8551164 0.80 DRD2 (0.53) DRD2SLC6A4HTR1DHTR1BSMN1; SMN2
SCHEMBL8702974 0.80 DRD2 (0.53) DRD2SLC6A4HTR1DHTR1BCHRM2
SCHEMBL8546639 0.79 SMN1; SMN2 (0.48) DRD2SLC6A4HTR1DHTR1BCHRM2
SCHEMBL8552288 0.79 DRD2 (0.43) DRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5792763-A MIGRAINES; ANALGESICS; DISEASES LINKED TO DECREASED NEUROTRANMISSION OF SEROTONIN IN MAMMALS ELI LILLY AND COMPANY (US) 1998-08-11 US disclosed
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed