SCHEMBL8553715

SCHEMBL8553715

NC(N)=Nc1nnc(-c2ccc(F)cc2)c2cccc(C(F)(F)F)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 6/20 0.38
NR1H3 Q13133 6/20 0.38
NR1I2 O75469 2/20 0.35
NR3C1 P04150 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 1/20 0.34
AR P10275 1/20 0.34
RXRA P19793 1/20 0.34
ESR1 P03372 3/20 0.33
PLAU P00749 2/20 0.33
ATP4A P20648 2/20 0.33
ATP4B P51164 2/20 0.33
PLG P00747 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552083 0.91 MEN1 (0.34) NR1H2NR1H3NR1I2NR3C1KDM4E
SCHEMBL8550323 0.90 PLG (0.42) NR1H2NR1H3KDM4EMEN1ALDH1A1
SCHEMBL8547668 0.89 PLAU (0.37) NR1H2NR1H3MEN1ALDH1A1HTT
Hydrochloric Acid SCHEMBL8548633 0.89 PLG (0.41) NR1H2NR1H3KDM4EMEN1ALDH1A1
SCHEMBL8546417 0.82 MEN1 (0.36) KDM4EMEN1ALDH1A1POLBHTT
SCHEMBL8554002 0.82 PLAU (0.44) KDM4EMEN1ALDH1A1POLBHTT
SCHEMBL8551154 0.81 CA9 (0.33) NR1H2NR1H3MAPTLMNASMN1; SMN2
SCHEMBL8551133 0.77 NR1H2 (0.42) NR1H2NR1H3NR1I2NR3C1MAPT
SCHEMBL8553708 0.76 LMNA (0.35) NR1H2NR1H3NR1I2NR3C1KDM4E
SCHEMBL8552274 0.74 PLAU (0.40) PLAUPLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed