SCHEMBL8556301

SCHEMBL8556301

O=C1NN(c2cccc(Cl)c2)C=C(Cl)C1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.46
HTT P42858 2/20 0.42
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
ADRB1 P08588 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTR1A P08908 1/20 0.42
CYP2D6 P10635 1/20 0.42
THRB P10828 1/20 0.42
CYP2C9 P11712 1/20 0.42
SLC6A4 P31645 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTR7 P34969 1/20 0.42
HTR3A P46098 1/20 0.42
HTR6 P50406 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4183804 0.85 GAA (0.39) ALOX5HTTGAAMEN1MAPT
SCHEMBL8557131 0.81 ALDH1A1 (0.43) HTTTP53ADRB1SLC6A4ALDH1A1
SCHEMBL10883345 0.75 ALDH1A1 (0.37) ALOX5HTTTP53THRBMGLL
SCHEMBL8554788 0.71 SIRT6 (0.42) TP53ADRB1ALDH1A1MEN1MAPT
SCHEMBL9645333 0.66 ALOX5 (0.45) ALOX5HTTHTR2AHTR2CHTR2B
SCHEMBL8751385 0.65 GAA (0.68) ALOX5HTTHTR2AHTR2CHTR2B
SCHEMBL19707986 0.64 MGLL (0.64) ALOX5HTTHTR2AHTR2CHTR2B
SCHEMBL3987095 0.63 ALOX5 (1.00) ALOX5ALDH1A1GAAMAPTHPGD
SCHEMBL11232168 0.63 ALOX5 (0.57) ALOX5HTTHTR2AHTR2CHTR2B
SCHEMBL11100857 0.63 ALDH1A1 (0.75) HTTHTR2AHTR2CHTR2BHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0756598-B1 SUBSTITUTED 5,6-DIHYDRO-5-OXO-1,4-DITHIINO-(2,3-D)-PYRIDAZINE-2,3-DICARBONITRILES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIALS DOW CHEMICAL CO (US) 1998-09-16 EP disclosed
EP-0756598-A1 SUBSTITUTED 5,6-DIHYDRO-5-OXO-1,4-DITHIINO-(2,3-D)-PYRIDAZINE-2,3-DICARBONITRILES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIALS THE DOW CHEMICAL COMPANY (a Delaware corporation) (US) 1997-02-05 EP disclosed
US-5488051-A BACTERICIDES, FUNGICIDES, ALGICIDES AND ANTIPROTOZOA AGENTS THE DOW CHEMICAL COMPANY (US) 1996-01-30 US disclosed
WO-1995029181-A1 SUBSTITUTED 5,6-DIHYDRO-5-OXO-1,4-DITHIINO-(2,3-D)-PYRIDAZINE-2,3-DICARBONITRILES, COMPOSITIONS CONTAINING THEM AND THEIR USE AS ANTIMICROBIALS THE DOW CHEMICAL COMPANY (US) 1995-11-02 WO disclosed