SCHEMBL8556983

SCHEMBL8556983

C=CCc1cc(CCC)c2c(c1O)C(C)(C)C(=O)N2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
GAA P10253 3/20 0.36
POLB P06746 2/20 0.36
KDM4E B2RXH2 3/20 0.35
PDK2 Q15119 1/20 0.35
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
GABRA1 P14867 1/20 0.32
GABRB2 P47870 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPK1 P28482 1/20 0.31
GLA P06280 1/20 0.30
ALOX5 P09917 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554202 0.93 MEN1 (0.35) DHFRMEN1KMT2AGAAPOLB
SCHEMBL8598630 0.91 MEN1 (0.34) MEN1KMT2AGAAPOLBKDM4E
SCHEMBL8556883 0.91 PDK2 (0.40) MEN1KMT2AGAAPOLBKDM4E
SCHEMBL8559143 0.90 GPR84 (0.36) MEN1KMT2AGAAPOLBKDM4E
SCHEMBL8560875 0.83 MEN1 (0.36) MEN1KMT2AGAAPOLBKDM4E
SCHEMBL8555558 0.71 GABRA1 (0.42) MEN1KMT2AGAAPOLBKDM4E
SCHEMBL8556960 0.71 PDK2 (0.44) PDK2ALOX5
SCHEMBL8560521 0.69 ALDH1A1 (0.35) GAAKDM4EHPGDALDH1A1GLA
SCHEMBL8560283 0.68 KDM4E (0.37) MEN1KMT2AGAAKDM4EPDK2
SCHEMBL8559665 0.68 PDK2 (0.33) PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653426-B1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA CO (JP) 1998-07-22 EP disclosed
EP-0653426-A1 Indole derivatives, salts thereof and heart affection therapeutic agent comprising the same KOWA COMPANY, LTD. (JP) 1995-05-17 EP disclosed