SCHEMBL8559867

SCHEMBL8559867

O=C(Nc1ccc(C(=O)N2c3ccccc3CNc3ccccc32)c(Cl)c1)c1ccccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.47
AVPR2 P30518 10/20 0.47
AVPR1A P37288 9/20 0.47
CHRM5 P08912 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
GRM4 Q14833 1/20 0.43
PKM P14618 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556908 0.93 RAB9A (0.47) RAB9AAVPR2AVPR1A
SCHEMBL8561432 0.93 AVPR2 (0.55) RAB9AAVPR2AVPR1A
SCHEMBL8561421 0.91 AVPR2 (0.56) AVPR2AVPR1AGRM4
SCHEMBL8556938 0.91 AVPR2 (0.56) AVPR2AVPR1AGRM4
SCHEMBL8564681 0.91 AVPR2 (0.42) AVPR2AVPR1A
SCHEMBL8557265 0.89 AVPR2 (0.58) RAB9AAVPR2AVPR1A
SCHEMBL8563330 0.89 NPC1 (0.47) RAB9AAVPR2AVPR1A
SCHEMBL8560617 0.88 AVPR1A (0.49) RAB9AAVPR2AVPR1AGRM4
SCHEMBL8561799 0.87 AVPR2 (0.59) RAB9AAVPR2AVPR1A
SCHEMBL8557787 0.86 PNLIP (0.50) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed