SCHEMBL8559038

SCHEMBL8559038

O=[N+]([O-])c1ccc2[nH]c(S(=O)(=O)Cc3ccccc3)nc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
MAPK1 P28482 1/20 0.53
CYP2C19 P33261 1/20 0.53
HIF1A Q16665 1/20 0.53
RIPK1 Q13546 2/20 0.50
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
MAPT P10636 3/20 0.47
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
NPBWR1 P48145 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HTT P42858 2/20 0.44
CYP19A1 P11511 1/20 0.43
GSR P00390 1/20 0.43
TXNRD1 Q16881 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559047 0.90 RIPK1 (0.62) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8554228 0.80 XDH (0.46) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7209149 0.79 ALDH1A1 (0.59) ALDH1A1MAPK1MAPTNPC1RAB9A
SCHEMBL10466630 0.78 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP3A4MEN1KMT2A
SCHEMBL16134487 0.78 L3MBTL1 (0.54) ALDH1A1CYP1A2CYP3A4RIPK1MEN1
SCHEMBL4006935 0.78 ALDH1A1 (0.51) ALDH1A1CYP3A4MEN1KMT2AMAPT
SCHEMBL6763997 0.77 RIPK1 (0.81) ALDH1A1RIPK1MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL6534097 0.77 ALDH1A1 (0.50) ALDH1A1CYP3A4MEN1KMT2AMAPT
SCHEMBL10465038 0.75 ALDH1A1 (0.46) ALDH1A1RIPK1MEN1KMT2AMAPT
SCHEMBL5504989 0.74 MAPT (0.73) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed