SCHEMBL8559047

SCHEMBL8559047

O=[N+]([O-])c1ccc2nc(S(=O)(=O)Cc3ccccc3)[nH]c2c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.62
MAPT P10636 6/20 0.56
NPBWR1 P48145 5/20 0.56
RAB9A P51151 4/20 0.56
NPC1 O15118 3/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
ALDH1A1 P00352 4/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
MAPK1 P28482 1/20 0.53
CYP2C19 P33261 1/20 0.53
HIF1A Q16665 1/20 0.53
L3MBTL1 Q9Y468 3/20 0.52
KDM4E B2RXH2 2/20 0.52
METAP1 P53582 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
GRIN1 Q05586 1/20 0.52
GRIN2B Q13224 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559038 0.90 ALDH1A1 (0.53) RIPK1MAPTNPBWR1RAB9ANPC1
SCHEMBL8554234 0.80 MAPT (0.56) MAPTRAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL7209149 0.79 ALDH1A1 (0.59) MAPTRAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL6773598 0.77 RIPK1 (1.00) RIPK1MAPTNPBWR1RAB9ANPC1
SCHEMBL8559255 0.74 MAPT (0.73) RIPK1MAPTNPBWR1RAB9ANPC1
SCHEMBL2245102 0.72 NPBWR1 (1.00) MAPTNPBWR1RAB9ANPC1SMN1; SMN2
SCHEMBL31679090 0.72 NPBWR1 (1.00) MAPTNPBWR1RAB9ANPC1SMN1; SMN2
SCHEMBL8554228 0.72 XDH (0.46) MAPTRAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL20380076 0.71 HTT (0.64) MAPTRAB9ANPC1ALDH1A1CYP1A2
SCHEMBL1171437 0.71 NPC1 (0.82) MAPTNPBWR1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0843671-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1998-05-27 EP disclosed
WO-1997003069-A1 HETEROCYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM GLAXO GROUP LIMITED (GB) 1997-01-30 WO disclosed