SCHEMBL8560767

SCHEMBL8560767

COC(=O)CCc1nc(NS(=O)(=O)c2ccccc2)c(-c2ccccc2)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 7/20 0.48
KDM4E B2RXH2 6/20 0.47
HPGD P15428 5/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
RXRA P19793 9/20 0.45
RXRB P28702 7/20 0.45
RXRG P48443 4/20 0.45
NR4A1 P22736 2/20 0.45
NR4A3 Q92570 2/20 0.45
TSHR P16473 2/20 0.45
MAPK1 P28482 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 2/20 0.45
ABCC4 O15439 1/20 0.45
C5 P01031 1/20 0.45
LMNA P02545 1/20 0.45
CHRM2 P08172 1/20 0.45
CHRM1 P11229 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560566 0.94 NR4A2 (0.47) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8560085 0.90 KDM4E (0.51) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8555950 0.89 TSHR (0.44) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8556747 0.89 RXRA (0.59) NR4A2KDM4EHPGDRXRARXRB
SCHEMBL8555804 0.84 TP53 (0.46) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8559306 0.84 RXRA (0.60) NR4A2KDM4EHPGDRXRARXRB
SCHEMBL8554937 0.83 MAPT (0.44) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8554882 0.83 NR4A2 (0.57) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8558225 0.82 NR4A2 (0.48) NR4A2KDM4EHPGDMEN1KMT2A
SCHEMBL8555034 0.81 ALDH1A1 (0.53) NR4A2KDM4EMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719163-A ARTHRITIS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed