Cyclamic Acid

Cyclamic Acid

SCHEMBL8563768

Cc1ncc(Cn2c(SC3CCNCC3)nc3ccccc32)o1.O=S(=O)(O)NC1CCCCC1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.43
MAPT P10636 3/20 0.37
GAA P10253 1/20 0.36
TSHR P16473 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LMNA P02545 2/20 0.35
HTT P42858 1/20 0.35
MC4R P32245 1/20 0.35
PPARG P37231 2/20 0.34
GSK3B P49841 1/20 0.34
PTAFR P25105 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
NR4A2 P43354 1/20 0.33
KCNH2 Q12809 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HIF1A Q16665 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfamic Acid Cyclohexyl Ester SCHEMBL9302699 0.85 MAPK1 (0.41) MAPK1MAPTTSHRMEN1KMT2A
Cyclamic Acid SCHEMBL9302048 0.78 KCNH2 (0.41) MAPTGAAMEN1KMT2ASMN1; SMN2
SCHEMBL8565877 0.74 HSD11B1 (0.46) MAPK1MAPTGAATSHRMEN1
Cyclamic Acid SCHEMBL8560203 0.74 KCNH2 (0.43) MAPTGAAMEN1KMT2ASMN1; SMN2
SCHEMBL8565135 0.73 GPR119 (0.42) MAPK1MAPTGAASMN1; SMN2MC4R
SCHEMBL9303969 0.73 KCNH2 (0.60) MAPTGAAMEN1KMT2ASMN1; SMN2
Cyclamic Acid SCHEMBL9303369 0.72 KCNH2 (0.40) MAPTGAAMEN1KMT2ASMN1; SMN2
SCHEMBL9537130 0.65 KCNH2 (0.63) MAPK1SMN1; SMN2LMNAMC4RNR4A2
SCHEMBL4991751 0.65 LMNA (0.45) MAPTTSHRMEN1KMT2ASMN1; SMN2
SCHEMBL14263834 0.65 TNF (0.57) MAPTTSHRSMN1; SMN2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0539421-B1 NOVEL OXAZOLYL DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 1998-09-23 EP disclosed
US-5278165-A Oxazolyl imidazol[4,5-b]pyridin and pyrimidine compounds JANSSEN PHARMACEUTICA N.V. (BE) 1994-01-11 US disclosed
US-5217980-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1993-06-08 US disclosed
EP-0539421-A1 NOVEL OXAZOLYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-05-05 EP disclosed
WO-1992001687-A1 NOVEL OXAZOLYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1992-02-06 WO disclosed