SCHEMBL8569833

SCHEMBL8569833

COc1ccc(Oc2ccccc2)cc1C(=O)CCCCCl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.48
HDAC8 Q9BY41 1/20 0.45
HDAC1 Q13547 1/20 0.45
KDM4E B2RXH2 2/20 0.45
POLB P06746 2/20 0.45
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
CAPN1 P07384 2/20 0.43
PPARG P37231 1/20 0.43
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
TTR P02766 2/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569807 0.87 KMT2A (0.53) HSD11B1HDAC8KDM4EPOLBMAPT
SCHEMBL8569681 0.82 HTR2A (0.56) HSD11B1HDAC8HDAC1KDM4EPOLB
SCHEMBL8572525 0.80 ALDH1A1 (0.56) HDAC8HDAC1KDM4EPOLBMEN1
SCHEMBL8569591 0.80 HDAC8 (0.67) HDAC8HDAC1KMT2ALMNAHTT
SCHEMBL8571105 0.79 HTR2A (0.55) POLBMAPTTSHRHTR2AHTR2C
SCHEMBL8572013 0.78 KDM4E (0.69) HSD11B1KDM4EPOLBMAPTTTR
SCHEMBL7261534 0.77 PDE4B (0.60) HSD11B1KDM4EMAPTTSHRCAPN1
SCHEMBL8567801 0.76 KCNK3 (0.55) KDM4EPOLBMAPTPPARGPPARA
SCHEMBL8571284 0.76 RAB9A (0.58) HDAC1POLBMAPTMEN1KMT2A
SCHEMBL7823697 0.76 PDE4B (0.62) HSD11B1KDM4EMAPTTSHRCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed