SCHEMBL8567801

SCHEMBL8567801

COc1ccc(NC(=O)c2ccccc2)cc1C(=O)CCCCCl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.55
KCNK9 Q9NPC2 1/20 0.55
KMT2A Q03164 6/20 0.51
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
MEN1 O00255 5/20 0.50
PPARG P37231 1/20 0.49
PPARA Q07869 1/20 0.49
NR1H4 Q96RI1 1/20 0.49
POLB P06746 1/20 0.49
MAPT P10636 3/20 0.47
MCHR1 Q99705 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
GRM5 P41594 1/20 0.47
RAB9A P51151 4/20 0.47
ALDH1A1 P00352 1/20 0.47
NPC1 O15118 2/20 0.47
NLRP3 Q96P20 1/20 0.47
ACHE P22303 1/20 0.47
SMO Q99835 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8570812 0.87 GRM4 (0.54) KCNK3KCNK9KMT2AKDM4EMEN1
SCHEMBL8574070 0.84 ALDH1A1 (0.51) KMT2AKDM4ELMNAMEN1POLB
SCHEMBL8570504 0.80 HTR6 (0.52) KMT2AKDM4ELMNAMEN1SMN1; SMN2
SCHEMBL8809240 0.80 GAA (0.59) LMNASMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL7050973 0.79 KCNK9 (0.67) KCNK3KCNK9KMT2AKDM4ELMNA
SCHEMBL8569681 0.78 HTR2A (0.56) KMT2AKDM4EMEN1NR1H4POLB
SCHEMBL8569833 0.76 HSD11B1 (0.48) KMT2AKDM4ELMNAMEN1PPARG
SCHEMBL8569591 0.76 HDAC8 (0.67) KMT2ALMNASMN1; SMN2RAB9AALDH1A1
SCHEMBL5492048 0.76 RAB9A (0.75) KCNK3KCNK9KMT2AKDM4EMEN1
SCHEMBL21357031 0.75 NPC1 (0.74) KMT2AKDM4ELMNAMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed