SCHEMBL8563393

SCHEMBL8563393

C=CCOC(=O)c1ccccc1Oc1cccc2c1C[C@@](NC(=O)OC(C)(C)C)(OC(=O)OC(C)(C)C)CC2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
GHSR Q92847 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KCNA3 P22001 2/20 0.33
CXCR5 P32302 2/20 0.33
RHOA P61586 1/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
LIG1 P18858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8573147 0.96 CYP3A4 (0.37) CYP3A4GHSRADRB2ADRB1ADRB3
SCHEMBL8845103 0.87 GHSR (0.41) CYP3A4GHSRADRB2ADRB1ADRB3
SCHEMBL8567143 0.84 CA1 (0.39) CYP3A4GHSRALDH1A1TSHR
SCHEMBL8575729 0.84 CA1 (0.39) CYP3A4GHSRALDH1A1TSHR
SCHEMBL8997625 0.78 GHSR (0.37) GHSRADRB2
SCHEMBL8569271 0.77 GHSR (0.39) GHSR
SCHEMBL8997648 0.77 SYK (0.38) GHSR
SCHEMBL8845155 0.76 GHSR (0.42) CYP3A4GHSRALDH1A1TSHRCXCR5
SCHEMBL8845267 0.76 GHSR (0.42) CYP3A4GHSRALDH1A1TSHRCXCR5
SCHEMBL8561422 0.76 CTSV (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640618-B1 Tetrahydronaphthalene-peptide derivatives HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed
EP-0640618-A1 Tetrahydronaphthalene-peptide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-03-01 EP disclosed