SCHEMBL8575779

SCHEMBL8575779

COc1ccc(N(S(=O)(=O)c2ccccc2)S(=O)(=O)c2ccccc2)cc1C(=O)CCCCCl

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.46
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
ABCB1 P08183 1/20 0.41
HDAC8 Q9BY41 1/20 0.40
HDAC1 Q13547 1/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPK1 P28482 1/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569681 0.79 HTR2A (0.56) HSD11B1KMT2AMEN1HDAC8HDAC1
SCHEMBL16540191 0.79 KMT2A (0.50) HSD11B1KMT2AMEN1ALDH1A1MAPK1
SCHEMBL8575784 0.79 HDAC3 (0.48) HSD11B1KMT2AMEN1HDAC8HDAC1
SCHEMBL8570504 0.78 HTR6 (0.52) HSD11B1KMT2AMEN1ALDH1A1MAPK1
SCHEMBL8569833 0.75 HSD11B1 (0.48) HSD11B1KMT2AMEN1HDAC8HDAC1
SCHEMBL31267400 0.74 ABCB1 (0.50) KMT2AMEN1ABCB1ALDH1A1MAPK1
SCHEMBL8569591 0.74 HDAC8 (0.67) KMT2AHDAC8HDAC1ALDH1A1
SCHEMBL8574314 0.74 HTR2C (0.60) KMT2AMEN1ALDH1A1HTR2AHTR2C
SCHEMBL8571105 0.73 HTR2A (0.55) KMT2AMEN1ALDH1A1MAPK1HTR2A
SCHEMBL8569807 0.73 KMT2A (0.53) HSD11B1KMT2AMEN1HDAC8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed