SCHEMBL8586535

SCHEMBL8586535

CCC(c1cc(S(=O)(=O)O)ccc1C)c1ccccc1F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
EEF2K O00418 3/20 0.38
CASR P41180 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TSHR P16473 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
PKM P14618 1/20 0.34
SNCA P37840 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28564255 0.83 LMNA (0.42) HTTTSHRCYP1A2CYP2C19SMN1; SMN2
SCHEMBL21274711 0.82 L3MBTL1 (0.39) HTTEEF2KCASRL3MBTL1TSHR
SCHEMBL7525829 0.76 HTT (0.33) HTTCYP1A2CYP2C19
SCHEMBL600325 0.76 ALDH1A1 (0.36) HTTCASRTSHRSNCA
SCHEMBL8813449 0.76 LMNA (0.43) HTTTSHRCYP2C19SMN1; SMN2SNCA
SCHEMBL9568576 0.75 HTT (0.38) HTTCASRTSHRCYP1A2CYP2C19
SCHEMBL776507 0.75 HTT (0.39) HTTCASRTSHRCYP1A2CYP2C19
SCHEMBL21910179 0.74 IDO1 (0.47) L3MBTL1TSHR
SCHEMBL9615906 0.74 HTT (0.43) HTTTSHRSNCA
SCHEMBL4687102 0.73 SLC6A2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0701546-B1 AROMATIC ACETYLCHOLINESTERASE INHIBITORS MERRELL PHARMA INC (US) 1998-12-23 EP disclosed
US-5663448-A Aromatic acetylcholinesterase inhibitors MERRELL PHARMACEUTICALS INC. (US) 1997-09-02 US disclosed
EP-0701546-A1 AROMATIC ACETYLCHOLINESTERASE INHIBITORS MERRELL PHARMACEUTICALS INC. (US) 1996-03-20 EP disclosed
WO-1994029255-A1 AROMATIC ACETYLCHOLINESTERASE INHIBITORS MERRELL PHARMACEUTICALS INC. (US) 1994-12-22 WO disclosed
EP-0627400-A1 Aromatic acetylcholinesterase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1994-12-07 EP disclosed