SCHEMBL8599745

SCHEMBL8599745

CCCCOC(=O)C(CC)N(C(C)=O)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.39
ATM Q13315 1/20 0.38
HPGD P15428 4/20 0.38
RAB9A P51151 4/20 0.38
ALDH1A1 P00352 4/20 0.38
L3MBTL1 Q9Y468 4/20 0.38
NPC1 O15118 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
LMNA P02545 3/20 0.37
TSHR P16473 3/20 0.37
MCL1 Q07820 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7576950 0.86 POLB (0.40) ESR1HPGDRAB9AALDH1A1L3MBTL1
SCHEMBL7404622 0.84 TSHR (0.39) HPGDALDH1A1L3MBTL1SMN1; SMN2TDP1
SCHEMBL7567342 0.82 CETP (0.40) HPGDRAB9AALDH1A1L3MBTL1NPC1
SCHEMBL7571120 0.81 ALDH1A1 (0.39) ESR1ATMHPGDRAB9AALDH1A1
SCHEMBL7569876 0.81 FAAH (0.39) ESR1HPGDRAB9AALDH1A1L3MBTL1
SCHEMBL7573230 0.81 TSHR (0.45) HPGDRAB9AALDH1A1L3MBTL1NPC1
SCHEMBL6136682 0.80 KMO (0.37) HPGDALDH1A1SMN1; SMN2LMNA
SCHEMBL7574293 0.80 LTB4R2 (0.40) HPGDRAB9AALDH1A1L3MBTL1NPC1
SCHEMBL7571050 0.80 LMNA (0.40) ESR1ATMHPGDRAB9AL3MBTL1
SCHEMBL7570565 0.80 ALDH1A1 (0.47) ESR1ATMHPGDRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0951464-A1 N-(ARYL/HETEROARYLACETYL) AMINO ACID ESTERS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING BETA-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS Elan Pharmaceuticals, Inc. (US) 1999-10-27 EP claimed
WO-1998022430-A9 N-(ARYL/HETEROARYLACETYL) AMINO ACID ESTERS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING b-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS 1998-08-20 WO claimed
WO-1998022430-A1 N-(ARYL/HETEROARYLACETYL) AMINO ACID ESTERS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING b-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1998-05-28 WO claimed