SCHEMBL8601552

SCHEMBL8601552

COc1cc(COc2cc(NC(C)=O)c(Cl)cc2C(Cl)CCCC=O)cc(OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 4/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
MTNR1B P49286 1/20 0.39
ENPP2 Q13822 1/20 0.36
BRD4 O60885 2/20 0.35
FGFR4 P22455 1/20 0.35
LMNA P02545 2/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
RORC P51449 1/20 0.34
MAPT P10636 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
GAA P10253 1/20 0.34
AGER Q15109 1/20 0.34
CNR1 P21554 1/20 0.33
PTPN1 P18031 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8600700 0.92 KDM4E (0.47) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8603828 0.87 MTNR1A (0.38) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8602614 0.86 AGER (0.40) KDM4EALDH1A1LMNAPOLBRORC
SCHEMBL8602051 0.80 MTNR1B (0.39) KDM4EALDH1A1MTNR1BBRD4MAPT
SCHEMBL7348962 0.72 ALDH1A1 (0.45) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL8970918 0.71 MTNR1B (0.43) KDM4EALDH1A1CYP1A2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL8602124 0.70 ENPP2 (0.35) ALDH1A1CYP2C19MTNR1BENPP2CYP3A4
SCHEMBL8971582 0.69 AGER (0.45) ALDH1A1LMNAPOLBMAPTMEN1
SCHEMBL8603248 0.69 ENPP2 (0.35) ALDH1A1CYP1A2CYP2C9CYP2C19ENPP2
SCHEMBL8602358 0.67 CYP3A4 (0.38) ALDH1A1CYP2C19ENPP2CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763458-A NERVOUS SYSTEM DISORDERS, ANXIETY, ANTIDEPRESSANTS AND COGNITION ACTIVATORS SYNTEX (U.S.A.) INC. (US) 1998-06-09 US disclosed