SCHEMBL8614302

SCHEMBL8614302

OC(CNCc1ccc(Cl)c(Cl)c1)CN1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.48
CACNA1G O43497 2/20 0.48
HTR2A P28223 7/20 0.47
DRD3 P35462 7/20 0.47
OPRK1 P41145 7/20 0.47
SLC6A3 Q01959 7/20 0.47
DRD5 P21918 6/20 0.47
HRH2 P25021 6/20 0.47
HTR7 P34969 6/20 0.47
OPRM1 P35372 6/20 0.47
HTR6 P50406 6/20 0.47
HRH1 P35367 6/20 0.47
OPRD1 P41143 6/20 0.47
DRD4 P21917 5/20 0.47
ADRA1D P25100 5/20 0.47
ADRA1A P35348 5/20 0.47
HTR1A P08908 4/20 0.47
CACNA1F O60840 4/20 0.47
ADRA1B P35368 4/20 0.47
CACNA1D Q01668 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8611835 0.89 DRD3 (0.49) KCNH2CACNA1GHTR2ADRD3OPRK1
SCHEMBL7751327 0.86 SLC6A3 (0.54) KCNH2HTR2ADRD3OPRK1SLC6A3
SCHEMBL8616693 0.85 HTR2A (0.50) KCNH2HTR2ADRD3OPRK1SLC6A3
Hydrochloric Acid SCHEMBL7544797 0.85 SLC6A3 (0.53) HTR2ADRD3OPRK1SLC6A3DRD5
SCHEMBL9416417 0.85 SLC6A3 (0.42) HTR2ADRD3OPRK1SLC6A3DRD5
SCHEMBL7754872 0.84 SLC6A3 (0.47) KCNH2CACNA1GHTR2ADRD3OPRK1
SCHEMBL9142370 0.83 KCNH2 (0.48) KCNH2CACNA1GHTR2ADRD3OPRK1
SCHEMBL8611930 0.83 MAPK1 (0.55) KCNH2HTR2ADRD3OPRK1SLC6A3
SCHEMBL9142194 0.80 MAPT (0.51) KCNH2CACNA1GHTR2ADRD3OPRK1
SCHEMBL9301460 0.78 CACNA1G (0.62) KCNH2CACNA1GHTR2ADRD3OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0549796-B1 DIPHENYLPIPERAZINE DERIVATIVE AND DRUG FOR CIRCULATORY ORGAN CONTAINING THE SAME POLA CHEM IND INC (JP) 1998-04-29 EP disclosed
US-5391552-A Has strong antagonism against calcium with less side effects POLA CHEMICAL INDUSTRIES, INC. (JP) 1995-02-21 US disclosed
EP-0612738-A1 Diphenylpiperazine derivative and drug for circulatory organ containing the same POLA CHEMICAL INDUSTRIES, INC. (JP) 1994-08-31 EP disclosed
EP-0549796-A1 DIPHENYLPIPERAZINE DERIVATIVE AND DRUG FOR CIRCULATORY ORGAN CONTAINING THE SAME POLA CHEMICAL INDUSTRIES INC (JP) 1993-07-07 EP disclosed