SCHEMBL8616047

SCHEMBL8616047

Cc1ccccc1-c1cc(NC(=N)NC=O)c2cc(NS(C)(=O)=O)ccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
LMNA P02545 3/20 0.45
HPGD P15428 3/20 0.45
HSP90AA1 P07900 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.45
NPSR1 Q6W5P4 2/20 0.45
THRB P10828 2/20 0.42
GAA P10253 1/20 0.42
MET P08581 5/20 0.41
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 1/20 0.40
KCNH2 Q12809 2/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CASP1 P29466 2/20 0.38
CASP7 P55210 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617771 0.93 ALDH1A1 (0.40) ALDH1A1LMNAHPGDHSP90AA1KDM4E
SCHEMBL8613743 0.88 ALDH1A1 (0.53) ALDH1A1LMNAHPGDHSP90AA1KDM4E
SCHEMBL8613752 0.87 KMT2A (0.42) ALDH1A1HPGDKDM4EMAPTTHRB
SCHEMBL8614948 0.84 HTT (0.39) ALDH1A1HPGDKDM4EMAPTGAA
SCHEMBL8620892 0.84 HTT (0.47) ALDH1A1HPGDKDM4EMAPTCYP1A2
SCHEMBL8617040 0.83 KEAP1 (0.41) HTTTP53
SCHEMBL8613761 0.82 TP53 (0.40) ALDH1A1LMNAHPGDHSP90AA1KDM4E
SCHEMBL8615149 0.82 ALDH1A1 (0.49) ALDH1A1LMNAHPGDHSP90AA1KDM4E
SCHEMBL8616673 0.82 CA2 (0.50) KDM4EMAPTCA2CA9CA12
SCHEMBL8615234 0.81 HTT (0.38) ALDH1A1HPGDKDM4EMAPTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed