SCHEMBL8625810

SCHEMBL8625810

CC(C)C(CC(N)=O)C(O)C(F)(F)C(=O)NCCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.44
OPRK1 P41145 1/20 0.44
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX12 P18054 1/20 0.43
MMP8 P22894 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
HPGD P15428 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
MLYCD O95822 2/20 0.41
EPHX1 P07099 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8761334 0.89 SMN1; SMN2 (0.40) POLBNPC1RAB9AALDH1A1CYP3A4
SCHEMBL8624798 0.87 SMN1; SMN2 (0.47) ALDH1A1KMT2AMEN1
SCHEMBL8762407 0.84 L3MBTL1 (0.49) NPC1RAB9AALDH1A1CYP2C19CYP1A2
SCHEMBL18228853 0.83 POLB (0.48) POLBOPRK1NPC1RAB9AALDH1A1
SCHEMBL21959109 0.83 POLB (0.48) POLBOPRK1NPC1RAB9AALDH1A1
SCHEMBL8627352 0.80 EPHX1 (0.34) EPHX1
SCHEMBL8627934 0.78 OPRK1 (0.44) POLBOPRK1NPC1RAB9AALDH1A1
SCHEMBL8762402 0.77 MAPK1 (0.44) POLBRAB9AALDH1A1CYP3A4MAPT
Hydrochloric Acid SCHEMBL7443223 0.71 OPRK1 (0.48) POLBOPRK1NPC1RAB9AALDH1A1
SCHEMBL3833319 0.70 MLYCD (0.62) POLBNPC1RAB9AALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636142-B1 LACTAM PEPTIDES HAVING HLE INHIBITING ACTIVITY ZENECA LTD (GB) 1998-06-17 EP disclosed
EP-0636141-B1 PYRIMIDINYL ACETAMIDES AS ELASTASE INHIBITORS ZENECA LTD (GB) 1997-06-25 EP disclosed