SCHEMBL8630486

SCHEMBL8630486

Cc1ncsc1C(O)c1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
ADRA2A P08913 5/20 0.44
ADRA2B P18089 5/20 0.44
ADRA2C P18825 5/20 0.44
ADRA1A P35348 4/20 0.44
ADRA1D P25100 3/20 0.44
ADRA1B P35368 3/20 0.44
TSHR P16473 1/20 0.44
GAA P10253 1/20 0.42
ALDH1A1 P00352 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CYP2A6 P11509 2/20 0.38
MAPT P10636 1/20 0.37
HSD17B10 Q99714 1/20 0.37
LTC4S Q16873 2/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629570 0.81 GAA (0.44) KMT2AGAAALDH1A1MAPTLMNA
SCHEMBL8629431 0.79 BRD4 (0.39)
SCHEMBL8633796 0.79 ADRB2 (0.36) CYP2C19
SCHEMBL8629520 0.78 ACHE (0.44) ALDH1A1CYP1A2MAPTLMNA
SCHEMBL2593085 0.74 SLC6A3 (0.44) ALDH1A1LMNA
SCHEMBL28036665 0.73 SLC6A4 (0.34) KMT2ATSHRGAAALDH1A1CYP1A2
SCHEMBL598905 0.73 ALDH1A1 (0.60) KMT2AADRA2AADRA2BADRA2CADRA1A
SCHEMBL31332147 0.73 ALDH1A1 (0.60) KMT2AADRA2AADRA2BADRA2CADRA1A
SCHEMBL9025658 0.70 IDO1 (0.38) MAPTLMNA
SCHEMBL8633347 0.69 TSHR (0.44) KMT2ATSHRALDH1A1MAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed