SCHEMBL8630535

SCHEMBL8630535

FC(F)(F)c1cccc(N2CCN(Cn3ncc4ccccc43)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.53
SMO Q99835 1/20 0.53
KDM4E B2RXH2 2/20 0.52
POLB P06746 1/20 0.52
DHFR P00374 2/20 0.52
SLC6A4 P31645 2/20 0.50
HTR2A P28223 1/20 0.50
ADRA1A P35348 3/20 0.49
DRD3 P35462 3/20 0.49
HTR1A P08908 2/20 0.49
ABCB11 O95342 1/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CHRM1 P11229 1/20 0.49
DRD1 P21728 1/20 0.49
TBXA2R P21731 1/20 0.49
OPRM1 P35372 1/20 0.49
KCNH2 Q12809 1/20 0.49
HTR7 P34969 1/20 0.49
DRD2 P14416 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8628212 0.91 SMO (0.42) SIGMAR1SMOKDM4EPOLBDHFR
SCHEMBL15748030 0.88 HTR2A (0.59) SIGMAR1SLC6A4HTR2AADRA1ADRD3
SCHEMBL8633681 0.83 RECQL (0.50) SIGMAR1SMOPOLBADRA1ADRD3
SCHEMBL8631540 0.82 KCNH2 (0.51) POLBDHFRHTR2ADRD3HTR1A
SCHEMBL8632193 0.82 KDM4E (0.52) KDM4EDRD3DRD1DRD2ALDH1A1
SCHEMBL8634968 0.80 DRD4 (0.57) SMOKDM4EPOLBALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL8629946 0.79 DRD4 (0.56) SMOKDM4EPOLBALDH1A1CYP1A2
SCHEMBL8629124 0.78 DRD4 (0.48) SLC6A4ADRA1ADRD3HTR1ADRD2
SCHEMBL8631570 0.76 MAPT (0.47) SMOKDM4EPOLBSLC6A4DRD3
SCHEMBL8629425 0.76 DRD4 (0.56) KDM4EPOLBADRA1ADRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed