SCHEMBL8634968

SCHEMBL8634968

FC(F)(F)c1ccc(N2CCN(Cn3ncc4ccccc43)CC2)nc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.57
GRM2 Q14416 1/20 0.57
HTT P42858 5/20 0.48
LMNA P02545 5/20 0.48
ALDH1A1 P00352 4/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
SMN1; SMN2 Q16637 8/20 0.46
SMO Q99835 2/20 0.46
MAPT P10636 5/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 3/20 0.45
TSHR P16473 2/20 0.45
HSD17B10 Q99714 2/20 0.45
USP2 O75604 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8629946 0.99 DRD4 (0.56) DRD4GRM2HTTLMNAALDH1A1
SCHEMBL8632193 0.84 KDM4E (0.52) DRD4GRM2LMNAALDH1A1MAPT
SCHEMBL8628029 0.82 DRD2 (0.46) DRD4GRM2L3MBTL1TSHRHSD17B10
SCHEMBL8630532 0.82 DRD2 (0.46) DRD4ALDH1A1KMT2AMAPTL3MBTL1
SCHEMBL8628212 0.81 SMO (0.42) DRD4GRM2SMOL3MBTL1KDM4E
SCHEMBL8628179 0.81 KDM4E (0.50) DRD4GRM2LMNAALDH1A1KMT2A
SCHEMBL8633168 0.80 HTR3A (0.55) LMNAALDH1A1MAPTL3MBTL1TSHR
SCHEMBL8630535 0.80 SIGMAR1 (0.53) ALDH1A1SMN1; SMN2SMOMAPTKDM4E
SCHEMBL8628045 0.80 DHFR (0.43) DRD4GRM2LMNAALDH1A1SMN1; SMN2
SCHEMBL8631634 0.77 HRH3 (0.59) HTTLMNAALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed