SCHEMBL8628212

SCHEMBL8628212

FC(F)(F)c1cc(N2CCN(Cn3ncc4ccccc43)CC2)cc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.42
DRD4 P21917 1/20 0.42
GRM2 Q14416 1/20 0.42
SIGMAR1 Q99720 2/20 0.41
DHFR P00374 1/20 0.41
SLC6A4 P31645 3/20 0.41
HTR2A P28223 1/20 0.41
POLB P06746 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ADRB1 P08588 1/20 0.40
ADRA1A P35348 2/20 0.39
DRD3 P35462 2/20 0.39
ABCB11 O95342 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
DRD1 P21728 1/20 0.39
TBXA2R P21731 1/20 0.39
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630535 0.91 SIGMAR1 (0.53) SMOSIGMAR1DHFRSLC6A4HTR2A
SCHEMBL8633681 0.82 RECQL (0.50) SMODRD4GRM2SIGMAR1POLB
SCHEMBL8632193 0.82 KDM4E (0.52) DRD4GRM2KDM4EADRB1DRD3
SCHEMBL8634968 0.81 DRD4 (0.57) SMODRD4GRM2POLBKDM4E
Hydrochloric Acid SCHEMBL8629946 0.81 DRD4 (0.56) SMODRD4GRM2POLBKDM4E
SCHEMBL8629124 0.80 DRD4 (0.48) DRD4SLC6A4ADRA1ADRD3HTR1A
SCHEMBL15748030 0.79 HTR2A (0.59) SIGMAR1SLC6A4HTR2AADRA1ADRD3
SCHEMBL8631570 0.78 MAPT (0.47) SMODRD4SLC6A4POLBKDM4E
SCHEMBL8629425 0.78 DRD4 (0.56) DRD4GRM2POLBKDM4EADRA1A
SCHEMBL8631540 0.77 KCNH2 (0.51) DRD4DHFRHTR2APOLBADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed