SCHEMBL8632193

SCHEMBL8632193

FC(F)(F)c1ccnc(N2CCN(Cn3ncc4ccccc43)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.52
L3MBTL1 Q9Y468 2/20 0.52
ADRB1 P08588 1/20 0.48
CYP2D6 P10635 1/20 0.47
LRRK2 Q5S007 1/20 0.43
ALDH1A1 P00352 3/20 0.42
LMNA P02545 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TRPV1 Q8NER1 2/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
DRD4 P21917 1/20 0.41
GRM2 Q14416 1/20 0.41
MAPT P10636 4/20 0.41
TSHR P16473 1/20 0.41
CXCR3 P49682 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD3 P35462 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634968 0.84 DRD4 (0.57) KDM4EL3MBTL1CYP2D6ALDH1A1LMNA
Hydrochloric Acid SCHEMBL8629946 0.83 DRD4 (0.56) KDM4EL3MBTL1CYP2D6ALDH1A1LMNA
SCHEMBL8630535 0.82 SIGMAR1 (0.53) KDM4ECYP2D6ALDH1A1MAPTTSHR
SCHEMBL8628212 0.82 SMO (0.42) KDM4EL3MBTL1ADRB1HSD17B10DRD4
SCHEMBL8628179 0.81 KDM4E (0.50) KDM4EALDH1A1LMNAHSD17B10DRD4
SCHEMBL8633168 0.80 HTR3A (0.55) L3MBTL1LRRK2ALDH1A1LMNAHSD17B10
SCHEMBL8627836 0.76 DRD4 (0.45) KDM4EL3MBTL1ALDH1A1LMNAHSD17B10
SCHEMBL8630532 0.74 DRD2 (0.46) L3MBTL1ALDH1A1HSD17B10TRPV1DRD4
SCHEMBL8628029 0.74 DRD2 (0.46) L3MBTL1HSD17B10PPARGPPARADRD4
SCHEMBL8633681 0.73 RECQL (0.50) L3MBTL1HSD17B10DRD4GRM2DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed