SCHEMBL8631464

SCHEMBL8631464

COc1ccc(-c2c(NS(=O)(=O)c3ccccc3)nn(CCc3ccccc3)c2COCc2ccccc2)cc1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 5/20 0.40
HTR6 P50406 1/20 0.38
KDR P35968 1/20 0.37
PTGS1 P23219 2/20 0.37
PTGS2 P35354 2/20 0.37
MAPT P10636 1/20 0.37
ADRB2 P07550 1/20 0.36
ADRB1 P08588 1/20 0.36
ADRB3 P13945 1/20 0.36
ERN1 O75460 1/20 0.36
ACLY P53396 1/20 0.36
TP53 P04637 1/20 0.36
MDM2 Q00987 1/20 0.36
PPARA Q07869 1/20 0.36
HTT P42858 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632160 0.92 CCR4 (0.41) PI4KBHTR6PTGS1PTGS2ERN1
SCHEMBL8632918 0.90 PI4KB (0.41) PI4KBHTR6KDRPTGS1PTGS2
SCHEMBL8634845 0.89 PI4KB (0.38) PI4KBHTR6PTGS1PTGS2ERN1
SCHEMBL8629870 0.89 NPC1 (0.39) PI4KBPTGS1PTGS2MAPTERN1
SCHEMBL8635623 0.87 PI4KB (0.44) PI4KBHTR6KDRPTGS1PTGS2
SCHEMBL8632809 0.85 PI4KB (0.42) PI4KBHTR6KDRPTGS1PTGS2
SCHEMBL8632227 0.84 GAA (0.43) PTGS2MAPT
SCHEMBL8634716 0.84 PI4KB (0.42) PI4KBHTR6KDRPTGS1PTGS2
SCHEMBL8631050 0.83 PTGS2 (0.42) PI4KBHTR6KDRPTGS1PTGS2
SCHEMBL7778127 0.82 PTGS2 (0.52) PI4KBPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed