SCHEMBL8633074

SCHEMBL8633074

CCc1cc(N(C)c2cccnc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2B6 P20813 1/20 0.37
CYP2C19 P33261 1/20 0.37
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
GRM5 P41594 3/20 0.36
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
POLQ O75417 1/20 0.34
HTT P42858 1/20 0.34
GRM2 Q14416 1/20 0.34
SYK P43405 1/20 0.34
LMNA P02545 1/20 0.33
KCNA5 P22460 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634555 0.87 MKNK1 (0.38) CYP3A4CYP2C9CYP2B6CYP2C19GAA
SCHEMBL8635757 0.86 SMN1; SMN2 (0.31) CYP3A4CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL8635203 0.86 HSP90AA1 (0.35) ALDH1A1TP53LMNA
SCHEMBL7768691 0.85 SLC9A1 (0.42)
SCHEMBL8633117 0.82 PDE4B (0.40) ALDH1A1MAPTHTTLMNA
SCHEMBL8631189 0.82 MEN1 (0.31)
SCHEMBL8635349 0.81 ALDH1A1 (0.39) ALDH1A1MAPTTSHRHTTLMNA
SCHEMBL8634504 0.81 FLT1 (0.38) CYP3A4CYP2C19HPGDALDH1A1MAPT
SCHEMBL8636231 0.80 MCL1 (0.33) ALDH1A1TP53MAPTHTTLMNA
SCHEMBL8635879 0.80 MTNR1A (0.43) CYP3A4CYP2C9CYP2C19ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed