SCHEMBL8635879

SCHEMBL8635879

CCc1cc(N(C)c2cccc(OC)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.43
MTNR1B P49286 10/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ESR1 P03372 1/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B2 P37059 2/20 0.37
HSD17B1 P14061 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632126 0.88 TUBB4A (0.37) ALDH1A1LMNA
SCHEMBL8635339 0.87 MTNR1A (0.42) MTNR1AMTNR1BESR1ALDH1A1LMNA
SCHEMBL8633117 0.86 PDE4B (0.40) ALDH1A1LMNA
SCHEMBL8635203 0.85 HSP90AA1 (0.35) ESR1ALDH1A1LMNA
SCHEMBL7764803 0.85 SLC9A1 (0.41)
SCHEMBL8635349 0.85 ALDH1A1 (0.39) ALDH1A1LMNA
SCHEMBL8633199 0.82 PER2 (0.36)
SCHEMBL8634165 0.81 ESR1 (0.39) NPSR1ESR1ALDH1A1
SCHEMBL8634504 0.80 FLT1 (0.38) ALDH1A1LMNACYP3A4CYP2D6ALOX15
SCHEMBL8633074 0.80 CYP3A4 (0.37) ALDH1A1LMNACYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed