SCHEMBL8633221

SCHEMBL8633221

N#CCn1nc(-c2ccccc2S(N)(=O)=O)c(-c2ccc(Cl)cc2)c1CO

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.38
PTGS1 P23219 2/20 0.38
F10 P00742 10/20 0.37
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
PRSS2 P07478 1/20 0.35
PRSS3 P35030 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633375 0.90 F10 (0.37) PTGS2F10F2PRSS1PRSS2
SCHEMBL8629795 0.87 PTGS2 (0.40) PTGS2PTGS1F10F2PRSS1
SCHEMBL8629956 0.86 PTGS2 (0.37) PTGS2PTGS1F10KDM4ECYP3A4
SCHEMBL8628758 0.86 HTR7 (0.40) PTGS2PTGS1F10CYP3A4CYP2C9
SCHEMBL8628708 0.86 PTGDR2 (0.38) PTGS2PTGS1F10F2PRSS1
SCHEMBL8632287 0.85 PTGS2 (0.42) PTGS2PTGS1KDM4ECYP3A4MAPT
SCHEMBL7777782 0.83 PTGS2 (0.50) PTGS2PTGS1CA1CA2CA4
SCHEMBL8635408 0.83 PTGS2 (0.36) PTGS2PTGS1F10KDM4ECYP3A4
SCHEMBL8631669 0.83 PTGES2 (0.38) PTGS2PTGS1F10F2PRSS1
SCHEMBL8631579 0.83 PTGS2 (0.42) PTGS2PTGS1F10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed