SCHEMBL8635172

SCHEMBL8635172

CCc1cc(Nc2ccccc2F)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.42
PSIP1 O75475 1/20 0.40
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.37
TYK2 P29597 5/20 0.36
JAK2 O60674 4/20 0.36
JAK1 P23458 4/20 0.36
JAK3 P52333 1/20 0.36
KIT P10721 1/20 0.36
STAT3 P40763 1/20 0.36
PDE4D Q08499 1/20 0.36
KCNH2 Q12809 1/20 0.36
PKM P14618 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634536 0.87 CXCL8 (0.43) CXCL8MAPTSMN1; SMN2ALDH1A1TYK2
SCHEMBL8631388 0.85 GAA (0.40) CXCL8MAPTSMN1; SMN2ALDH1A1ALOX15
SCHEMBL8633397 0.85 AKR1C3 (0.43) MAPTSMN1; SMN2ALDH1A1TSHRNPC1
SCHEMBL8635140 0.84 BCAT2 (0.42) MAPTALDH1A1ALOX15GAAMEN1
SCHEMBL8636186 0.84 AKR1C3 (0.44) MAPTSMN1; SMN2ALDH1A1TSHRNPC1
SCHEMBL7768639 0.83 SLC9A1 (0.45)
SCHEMBL8633057 0.83 L3MBTL1 (0.41) ALDH1A1ALOX15TSHRGAALMNA
SCHEMBL8635300 0.82 HTT (0.38) MAPTALDH1A1HTT
SCHEMBL8632359 0.81 MEN1 (0.44) MAPTSMN1; SMN2GAARAB9AHTT
SCHEMBL8635911 0.79 TYK2 (0.47) SMN1; SMN2TSHRTYK2JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed