SCHEMBL8636968

SCHEMBL8636968

CC(=O)N(N1CCN(c2ccncc2)CC1)S(=O)(=O)CCCCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.45
SLC6A4 P31645 1/20 0.45
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
RORC P51449 6/20 0.40
SIGMAR1 Q99720 2/20 0.40
HTR1A P08908 2/20 0.40
DRD2 P14416 2/20 0.40
RORB Q92753 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636978 0.72 ITGB3 (0.41) RORC
SCHEMBL8634088 0.71 ITGB3 (0.36) RORC
SCHEMBL8635262 0.68 ITGB3 (0.48)
SCHEMBL8632400 0.67 MEN1 (0.39) RORCHTR1ADRD2
SCHEMBL8634075 0.67 RORC (0.45) RORCRORB
SCHEMBL7493712 0.66 DRD4 (0.61) DRD4SLC6A4HTR2AHTR1ADRD2
SCHEMBL8632726 0.65 KHK (0.44) DRD4RORC
SCHEMBL7403454 0.65 DRD4 (0.59) DRD4SLC6A4HTR1ADRD2
SCHEMBL12261943 0.64 DRD4 (0.77) DRD4HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8699932 0.63 GAA (0.42) HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed