SCHEMBL8636978

SCHEMBL8636978

CCCC(c1ccccc1)S(=O)(=O)N(C(C)=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.41
ITGA2B P08514 3/20 0.41
RORC P51449 2/20 0.38
KDM4E B2RXH2 3/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
CHRM1 P11229 2/20 0.37
TSHR P16473 1/20 0.36
SPHK1 Q9NYA1 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633916 0.75 ADRB2 (0.35) ITGB3ITGA2BCHRM1
SCHEMBL8634088 0.75 ITGB3 (0.36) ITGB3ITGA2BRORCKDM4EGAA
SCHEMBL8636968 0.72 DRD4 (0.45) RORC
SCHEMBL8634075 0.72 RORC (0.45) RORC
SCHEMBL8636260 0.71 SPHK1 (0.35) ITGB3ITGA2BRORCCHRM1TSHR
SCHEMBL8636258 0.67 OPRM1 (0.36) ITGB3ITGA2BRORCCHRM1SPHK1
Hydrochloric Acid SCHEMBL8837964 0.66 ITGB3 (0.45) ITGB3ITGA2BTSHRCYP2C9
SCHEMBL7400370 0.65 PPARG (0.50) ITGB3ITGA2BTSHRSPHK1CYP2C9
SCHEMBL8635262 0.65 ITGB3 (0.48) ITGB3ITGA2BKDM4EMAPTTSHR
SCHEMBL8636975 0.63 ITGB3 (0.39) ITGB3ITGA2BKDM4EGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed