SCHEMBL8637032

SCHEMBL8637032

CCc1cc(N(C)c2ccccn2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
HSD17B10 Q99714 1/20 0.34
POLB P06746 2/20 0.34
BRD4 O60885 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
MAPT P10636 1/20 0.33
THRB P10828 1/20 0.33
POLQ O75417 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
JAK2 O60674 1/20 0.31
KIT P10721 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631189 0.87 MEN1 (0.31) KMT2AMEN1HSD17B10
SCHEMBL8634361 0.86 BRD4 (0.39) ALDH1A1KMT2AMEN1HSD17B10POLB
SCHEMBL27351468 0.86 HRH4 (0.37)
SCHEMBL7766532 0.84 SLC9A1 (0.43)
SCHEMBL8635203 0.82 HSP90AA1 (0.35) ALDH1A1KMT2AMEN1POLBTHRB
SCHEMBL8634234 0.81 MEN1 (0.36) KMT2AMEN1HSD17B10POLB
SCHEMBL8635757 0.81 SMN1; SMN2 (0.31) ALDH1A1MAPTPOLQCYP2D6CYP2C19
SCHEMBL8635259 0.81 ALDH1A1 (0.38) ALDH1A1KMT2ATHRB
SCHEMBL8635336 0.80 FFAR2 (0.33)
SCHEMBL8633074 0.79 CYP3A4 (0.37) ALDH1A1MAPTPOLQCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1057999-C 4-Aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed
CN-1138575-A 4-aminobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-12-25 CN disclosed