SCHEMBL8395334

SCHEMBL8395334

COc1cccc(Oc2c(Cl)nc(-c3ccco3)nc2OS(=O)(=O)c2ccc(C(C)C)cn2)c1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
EDNRA P25101 9/20 0.36
NPBWR1 P48145 3/20 0.35
MCHR1 Q99705 3/20 0.35
PTGER4 P35408 1/20 0.35
DHPS P49366 1/20 0.33
EDNRB P24530 8/20 0.33
MAPT P10636 1/20 0.33
PIN1 Q13526 1/20 0.33
ADORA3 P0DMS8 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8398581 0.89 NPBWR1 (0.35) EDNRANPBWR1MCHR1DHPSEDNRB
SCHEMBL8398732 0.88 EDNRA (0.42) LMNAEDNRADHPSEDNRB
SCHEMBL7589754 0.85 EDNRA (0.47) EDNRAEDNRB
SCHEMBL8398843 0.77 DHPS (0.41) EDNRADHPSEDNRBADORA3ADORA2A
SCHEMBL7591710 0.76 EDNRA (0.56) EDNRAEDNRB
SCHEMBL8635722 0.76 DHPS (0.35) EDNRANPBWR1MCHR1DHPSEDNRB
SCHEMBL7589698 0.76 ALDH1A1 (0.47) DHPSMAPTADORA3ADORA2AADORA1
SCHEMBL7580836 0.74 EDNRA (0.44) EDNRAEDNRB
SCHEMBL8637899 0.73 DHPS (0.43) EDNRADHPSEDNRB
SCHEMBL7991567 0.71 EDNRA (0.62) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856484-A Sulfonylaminopyrimidine carboxylic acid derivatives having endothelin inhibiting activity HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed