SCHEMBL8638141

SCHEMBL8638141

Clc1ccc([C]2CCNC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.52
HTR2C P28335 5/20 0.50
SOS1 Q07889 1/20 0.49
PNMT P11086 3/20 0.47
ASIC3 Q9UHC3 1/20 0.44
HTR2A P28223 4/20 0.43
HTR2B P41595 4/20 0.43
HTR7 P34969 3/20 0.43
HTR6 P50406 2/20 0.43
HTR3A P46098 1/20 0.43
HTR1D P28221 1/20 0.42
HTR1E P28566 1/20 0.42
SLC2A1 P11166 1/20 0.38
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
LMNA P02545 1/20 0.37
RECQL P46063 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27926376 0.86 SIGMAR1 (0.55) SIGMAR1HTR2CSOS1PNMTASIC3
SCHEMBL8635851 0.78 HTR2A (0.42) HTR2CHTR2AHTR2BHTR7HTR6
SCHEMBL8350829 0.78 AHR (0.48) HTR2CPNMTASIC3HTR2AHTR2B
SCHEMBL27676378 0.77 PRCP (0.48) SIGMAR1HTR2CPNMTHTR7
SCHEMBL8639724 0.76 HTR2C (0.56) SIGMAR1HTR2CPNMTASIC3HTR2A
SCHEMBL3741829 0.74 PKN2 (0.50) PNMTLMNA
SCHEMBL8638940 0.74 NISCH (0.43) SIGMAR1HTR2CHTR2AHTR2BHTR7
SCHEMBL8355638 0.74 ASIC3 (0.46) HTR2CASIC3HTR2AHTR2B
SCHEMBL315185 0.73 LMNA (0.50) SIGMAR1HTR2CLMNARECQL
SCHEMBL8323150 0.71 ASIC3 (0.78) HTR2CPNMTASIC3HTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104114543-A Therapeutically active compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2014-10-22 CN claimed
CN-104114543-A Therapeutically active compounds and methods of use thereof AGIOS PHARMACEUTICALS INC 2014-10-22 CN disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed