SCHEMBL8639136

SCHEMBL8639136

CCN1CCCC1Oc1ccc(Cc2ccccc2)cc1C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
CRHBP P24387 2/20 0.42
CRHR2 Q13324 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.41
LTA4H P09960 5/20 0.40
CD274 Q9NZQ7 7/20 0.39
PDCD1 Q15116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637439 0.87 LTA4H (0.50) SMN1; SMN2ALDH1A1LTA4HCD274PDCD1
SCHEMBL8638836 0.85 KDM4E (0.38) SMN1; SMN2CRHBPCRHR2ALDH1A1MAPT
SCHEMBL8637725 0.82 CRHBP (0.38) SMN1; SMN2CRHBPCRHR2ALDH1A1MAPT
SCHEMBL8641866 0.82 LTA4H (0.42) SMN1; SMN2LTA4HCD274
SCHEMBL8637445 0.79 HRH1 (0.46) LTA4H
SCHEMBL8638274 0.77 LTA4H (0.39) LTA4H
SCHEMBL8637775 0.75 MAOA (0.44) SMN1; SMN2ALDH1A1LTA4H
SCHEMBL8638269 0.75 LTA4H (0.50) LTA4H
SCHEMBL8641109 0.75 LTA4H (0.52) ALDH1A1LTA4H
SCHEMBL8641764 0.75 HRH3 (0.50) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed