SCHEMBL8662809

SCHEMBL8662809

COc1ccccc1C(OCC1CC(O)CN1C(=O)c1cccn1C)(c1ccccc1)c1ccccc1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.37
CYP3A4 P08684 3/20 0.35
ALDH1A1 P00352 1/20 0.35
PDE4B Q07343 1/20 0.34
SLC6A1 P30531 3/20 0.33
KMT2A Q03164 2/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
SLC6A11 P48066 1/20 0.32
RIPK1 Q13546 1/20 0.31
CYP2C19 P33261 1/20 0.31
PIK3CD O00329 1/20 0.31
PABPC1 P11940 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ABCB1 P08183 1/20 0.31
HTT P42858 1/20 0.31
ITGB2 P05107 1/20 0.31
ICAM1 P05362 1/20 0.31
ITGAL P20701 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662816 0.92 CYP2D6 (0.36) CYP2D6CYP3A4ALDH1A1PDE4BSLC6A1
SCHEMBL8660375 0.86 SLC6A1 (0.36) SLC6A1KMT2ASLC6A11RIPK1PIK3CD
SCHEMBL8662093 0.82 PIK3CD (0.35) SLC6A1KMT2ASLC6A11RIPK1PIK3CD
SCHEMBL8662709 0.82 MTNR1B (0.37) SLC6A1KMT2ASLC6A11RIPK1HTT
SCHEMBL6858148 0.81 ITGA4 (0.39) KMT2AMEN1TP53
SCHEMBL8662962 0.81 PIK3CD (0.47) CYP2D6CYP3A4ALDH1A1KMT2APIK3CD
SCHEMBL8660410 0.80 POLB (0.44) CYP2D6CYP3A4ALDH1A1PDE4BKMT2A
SCHEMBL8661342 0.79 ALDH1A1 (0.35) CYP3A4ALDH1A1SLC6A1KMT2ACYP2C19
SCHEMBL8662486 0.79 MTNR1B (0.40) KMT2ASMN1; SMN2MEN1
SCHEMBL8662934 0.78 SLC6A1 (0.33) SLC6A1SLC6A11RIPK1HTTITGB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5714606-A OLIGONUCLEOTIDE HAVING RECEPTOR BINDING SITES; ENZYME INHIBITORS, ANTIINFLAMMATORY AGENTS, MEDICAL DIAGNOSIS ISIS PHARMACEUTICALS, INC. (US) 1998-02-03 US disclosed
EP-0739335-A4 PYRROLIDINE-CONTAINING MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS INC (US) 1997-04-02 EP disclosed
EP-0739335-A1 PYRROLIDINE-CONTAINING MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 1996-10-30 EP disclosed
WO-1995018792-A1 PYRROLIDINE-CONTAINING MONOMERS AND OLIGOMERS ISIS PHARMACEUTICALS, INC. (US) 1995-07-13 WO disclosed