SCHEMBL8664507

SCHEMBL8664507

FC(F)(F)c1cc[c]c(-c2ccccc2N2CCOCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 4/20 0.49
LMNA P02545 3/20 0.49
MAPT P10636 4/20 0.43
GAA P10253 2/20 0.43
PRKDC P78527 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TSHR P16473 3/20 0.39
HSD17B10 Q99714 2/20 0.39
CNR2 P34972 1/20 0.39
AKR1C3 P42330 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
ALOX15 P16050 1/20 0.38
AGER Q15109 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997939 0.83 L3MBTL1 (0.43) ALDH1A1LMNAMAPTGAAPRKDC
SCHEMBL8666713 0.80 MAPT (0.43) ALDH1A1LMNAMAPTGAAPRKDC
SCHEMBL8665551 0.80 MEN1 (0.43) ALDH1A1LMNAMAPTPRKDCL3MBTL1
SCHEMBL8663214 0.77 MAPT (0.40) ALDH1A1KDM4ELMNAMAPTL3MBTL1
SCHEMBL8667066 0.75 ALDH1A1 (0.49) ALDH1A1KDM4ELMNAMAPTKMT2A
SCHEMBL8665467 0.72 ALDH1A1 (0.55) ALDH1A1KDM4EMAPTGAAL3MBTL1
SCHEMBL2432403 0.71 GPR3 (0.41) ALDH1A1TSHR
SCHEMBL5778162 0.71 HSD11B1 (0.38) ALDH1A1TSHR
SCHEMBL8416356 0.70 HSD11B1 (0.42)
SCHEMBL4287156 0.69 ALDH1A1 (0.44) ALDH1A1KDM4ELMNAMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852006-A N-aminoalkyl-substituted nitrogen-containing six membered heterocyclic compounds NIPPON CHEMIPHAR CO., LTD. (JP) 1998-12-22 US disclosed
US-5574030-A INHIBITING URINARY CONTRACTION, HETEROCYCLIC DIAMINES NIPPON CHEMIPHAR CO., LTD. (JP) 1996-11-12 US disclosed