SCHEMBL8664656

SCHEMBL8664656

CC(=O)OCc1cc(Br)ccc1-n1c(Cl)nn(C)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SETDB1 Q15047 1/20 0.40
ALDH1A1 P00352 1/20 0.38
PTGER1 P34995 7/20 0.35
UCHL1 P09936 2/20 0.35
UCHL3 P15374 2/20 0.35
CASP2 P42575 1/20 0.33
CUL4A Q13619 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP1A2 P05177 2/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664792 0.88 SETDB1 (0.42) SETDB1ALDH1A1PTGER1UCHL1UCHL3
SCHEMBL8663188 0.87 ALDH1A1 (0.42) SETDB1ALDH1A1SMN1; SMN2CYP2C19CYP1A2
SCHEMBL8667576 0.83 ALDH1A1 (0.39) SETDB1ALDH1A1SMN1; SMN2CYP2C19CYP2C9
SCHEMBL8675983 0.81 SETDB1 (0.38) SETDB1ALDH1A1PTGER1CASP2CUL4A
SCHEMBL23712860 0.72 P2RX7 (0.35) CASP2SMN1; SMN2MEN1KMT2A
SCHEMBL28049660 0.69 ALDH1A1 (0.43) ALDH1A1CYP2C9CYP1A2MEN1KMT2A
SCHEMBL8670561 0.69 DDR1 (0.35) SETDB1ALDH1A1SMN1; SMN2CYP2C19CYP1A2
SCHEMBL21713935 0.68 FFAR4 (0.44) SETDB1ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL8664609 0.67 SETDB1 (0.37) SETDB1SMN1; SMN2MEN1KMT2A
SCHEMBL18498771 0.67 KDM4E (0.43) ALDH1A1SMN1; SMN2CYP2C19CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0874831-A1 PROCESSES AND COMPOUNDS FOR PREPARING CYCLIC UREA FUNGICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-11-04 EP disclosed
WO-1997019935-A1 PROCESSES AND COMPOUNDS FOR PREPARING CYCLIC UREA FUNGICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1997-06-05 WO disclosed