SCHEMBL8699355

SCHEMBL8699355

CCc1cc(NC(=O)N2CCN(c3ccccc3F)CC2C)c(OC)nc1C

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.45
RBP4 P02753 1/20 0.44
ROCK2 O75116 6/20 0.43
PRKG1 Q13976 6/20 0.43
CYP1A2 P05177 3/20 0.43
LIMK2 P53671 1/20 0.43
MAPT P10636 2/20 0.43
KMT2A Q03164 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 1/20 0.43
MEN1 O00255 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
PANK3 Q9H999 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8701411 0.90 TACR3 (0.47) RBP4ROCK2PRKG1MAPTKMT2A
SCHEMBL8704636 0.86 KMT2A (0.57) RBP4CYP1A2MAPTKMT2ANPSR1
SCHEMBL8700086 0.83 RBP4 (0.47) CHRM4RBP4ROCK2PRKG1LIMK2
SCHEMBL8699351 0.80 ALDH1A1 (0.66) CYP1A2MAPTKMT2ANPSR1ALDH1A1
SCHEMBL8701044 0.79 KMT2A (0.65) CYP1A2MAPTKMT2ANPSR1ALDH1A1
SCHEMBL8702850 0.78 PANK3 (0.56) MAPTKMT2ANPSR1ALDH1A1LMNA
SCHEMBL8701100 0.77 MAPT (0.39) MAPTKMT2AALDH1A1LMNATSHR
SCHEMBL8705064 0.76 HTR1A (0.52) RBP4MAPTKMT2ANPSR1ALDH1A1
SCHEMBL8699098 0.76 PANK3 (0.54) RBP4CYP1A2MAPTKMT2ANPSR1
SCHEMBL8704639 0.76 ALDH1A1 (0.40) CYP1A2MAPTKMT2ANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780472-A ANTITUMOR AGENTS SAMJIN PHARMACEUTICAZL CO., LTD. (KR) 1998-07-14 US disclosed