SCHEMBL8700409

SCHEMBL8700409

COC(=O)c1cc(S(C)(=O)=O)c(-c2ccccn2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 5/20 0.44
JAK1 P23458 2/20 0.43
TYK2 P29597 2/20 0.43
AXL P30530 1/20 0.43
SDHB P21912 1/20 0.42
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
SLC6A3 Q01959 2/20 0.41
ALB P02768 1/20 0.41
HTR1A P08908 1/20 0.41
SLC6A2 P23975 1/20 0.41
PDE4A P27815 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41
HTR2B P41595 1/20 0.41
PDE4D Q08499 1/20 0.41
SHH Q15465 1/20 0.41
USP28 Q96RU2 1/20 0.41
SLC29A1 Q99808 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8704331 0.86 SLC6A3 (0.50) JAK1TYK2AXLSDHBGABRG2
SCHEMBL8447990 0.81 SLC9A1 (0.47)
SCHEMBL8894494 0.79 PTGS2 (0.49) JAK1TYK2GRM5GAAMAPT
SCHEMBL8704080 0.79 CFTR (0.50) GABRG2GABRB3GABRA3LMNA
SCHEMBL205611 0.75 AXL (0.57) KAT6AAXLGABRG2GABRB3GABRA3
SCHEMBL17239550 0.74 NTRK1 (0.53)
SCHEMBL29694130 0.73 SLC6A3 (0.55) AXLSDHBGABRG2GABRB3GABRA3
SCHEMBL5234641 0.73 SLC6A3 (0.55) AXLSDHBGABRG2GABRB3GABRA3
SCHEMBL8700008 0.73 GABRG2 (0.43) JAK1TYK2AXLSDHBGABRG2
SCHEMBL3551797 0.73 SLC6A3 (0.52) KAT6AAXLGABRG2GABRB3GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753680-A Heterocyclyl-benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-19 US disclosed