SCHEMBL8894494

SCHEMBL8894494

COC(=O)c1ccc(-c2ccccn2)c(S(C)(=O)=O)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.49
VCAM1 P19320 1/20 0.46
JAK1 P23458 2/20 0.46
TYK2 P29597 2/20 0.46
ALOX15 P16050 1/20 0.46
HTT P42858 1/20 0.46
TGFBR1 P36897 1/20 0.46
KDM4E B2RXH2 4/20 0.45
KDM6B O15054 1/20 0.45
KDM5C P41229 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
KDM2A Q9Y2K7 1/20 0.45
KDM3A Q9Y4C1 1/20 0.45
GRM5 P41594 1/20 0.44
POLB P06746 2/20 0.44
MAPT P10636 1/20 0.44
CMA1 P23946 1/20 0.43
PKM P14618 2/20 0.42
ALDH1A1 P00352 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14886606 0.81 ALOX15 (0.50) ALOX15HTTTGFBR1KDM4EKDM6B
SCHEMBL5831775 0.80 ADORA3 (0.51) ALOX15HTTTGFBR1KDM4EKDM6B
SCHEMBL14886809 0.80 ALOX15 (0.49) ALOX15HTTTGFBR1KDM4EKDM6B
SCHEMBL8700409 0.79 KAT6A (0.44) JAK1TYK2GRM5MAPTGAA
SCHEMBL8704331 0.79 SLC6A3 (0.50) PTGS2JAK1TYK2GRM5MAPT
Hydrochloric Acid SCHEMBL8894574 0.79 JAK1 (0.41) JAK1TYK2KDM4EKDM5CALDH1A1
SCHEMBL13117413 0.79 ALOX15 (0.50) ALOX15HTTTGFBR1KDM4EKDM6B
SCHEMBL22636873 0.78 ALPL (0.52) PTGS2KDM4EPOLBMAPTALDH1A1
SCHEMBL22636820 0.78 PTGS2 (0.44) PTGS2JAK1TYK2TGFBR1KDM4E
SCHEMBL29430653 0.78 ALPL (0.52) PTGS2KDM4EPOLBMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693672-A 3,4,5-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-02 US disclosed