SCHEMBL8705122

SCHEMBL8705122

O=C(NS(=O)(=O)c1ccccc1)C(Cc1cccc(NS(=O)(=O)c2ccccc2)c1)c1ccc2nsnc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 6/20 0.45
PTGES O14684 1/20 0.43
PKLR P30613 1/20 0.42
ITGB3 P05106 1/20 0.41
ITGAV P06756 1/20 0.41
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
IKBKB O14920 1/20 0.39
PHGDH O43175 2/20 0.38
HDAC1 Q13547 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
AURKA O14965 1/20 0.38
RPS6KB1 P23443 1/20 0.38
PFKFB3 Q16875 1/20 0.38
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705444 0.95 PTGES (0.43) HTR6PTGESPKLRITGB3ITGAV
SCHEMBL8709447 0.90 ITGB3 (0.48) PKLRITGB3ITGAVMAPTMEN1
SCHEMBL8709683 0.89 ITGB3 (0.43) PKLRITGB3ITGAVMAPTKDM4E
SCHEMBL8712032 0.84 SLC7A5 (0.43) ITGB3ITGAVMAPTMEN1KMT2A
SCHEMBL8707148 0.83 KDM4E (0.43) ITGB3ITGAVMAPTKDM4EMEN1
SCHEMBL8705462 0.83 MAPT (0.44) PKLRITGB3ITGAVMAPTMEN1
SCHEMBL8709540 0.83 ITGB3 (0.43) ITGB3ITGAVMEN1KMT2APOLB
SCHEMBL8705691 0.82 MAPT (0.50) ITGB3ITGAVMAPTMEN1KMT2A
SCHEMBL8711591 0.81 ITGB3 (0.38) PKLRITGB3ITGAVMAPTKDM4E
SCHEMBL8709162 0.81 MAPT (0.45) ITGB3ITGAVMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998041515-A1 ENDOTHOLIN RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-09-24 WO disclosed