Camostat

Camostat

SCHEMBL871583

CN(C)C(=O)COC(=O)Cc1ccc(OC(=O)c2ccc(NC(=N)N)cc2)cc1.CS(=O)(=O)O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of Camostat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 known ✓ P00734 4/20 0.72
ADRA1A known ✓ P35348 1/20 0.63
PRSS1 P07477 6/20 0.72
KLK1 P06870 5/20 0.72
SLC22A2 O15244 1/20 0.63
TMPRSS2 O15393 1/20 0.63
HPN P05981 1/20 0.63
PRSS2 P07478 1/20 0.63
CTSL P07711 1/20 0.63
CNR1 P21554 1/20 0.63
PRSS3 P35030 1/20 0.63
OPRD1 P41143 1/20 0.63
HGFAC Q04756 1/20 0.63
KCNH2 Q12809 1/20 0.63
SLC47A2 Q86VL8 1/20 0.63
SLC47A1 Q96FL8 1/20 0.63
KLK7 P49862 4/20 0.43
POLB P06746 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Camostat SCHEMBL125269 0.96 PRSS1 (0.68) PRSS1KLK1F2SLC22A2TMPRSS2
SCHEMBL20008640 0.96 PRSS1 (0.68) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL2782237 0.95 PRSS1 (0.67) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL8829828 0.94 PRSS1 (0.66) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL1645380 0.93 PRSS1 (0.64) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL1645520 0.92 PRSS1 (0.63) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL23803656 0.91 PRSS1 (0.62) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL1646099 0.91 PRSS1 (0.62) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL1648303 0.91 PRSS1 (0.62) PRSS1KLK1F2SLC22A2TMPRSS2
Camostat SCHEMBL2326660 0.91 PRSS1 (0.62) PRSS1KLK1F2SLC22A2TMPRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1684 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS CENTRE FOR DIGESTIVE DISEASES (AU) 2026-05-21 US claimed
WO-2026089565-A1 USE OF CATHEPSIN L INHIBITOR IN COMBINATION ADMINISTRATION 연세대학교 산학협력단 2026-04-30 WO claimed
US-12458622-B2 Methods of treatment of coronavirus-induced inflammation conditions THE GENERAL HOSPITAL CORPORATION (US) 2025-11-04 US claimed
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2025-06-12 US claimed
US-20250152748-A1 HYDRODYNAMIC GENE DELIVERY UNIV JOHNS HOPKINS (US) 2025-05-15 US claimed
WO-2025097070-A1 ORAL DOSAGE FORM WITH CATIONICALLY CHARGEABLE HYDROGEL FOR DELIVERY OF ACTIVE AGENT ENTREGA INC. (US) 2025-05-08 WO claimed
WO-2025097068-A1 ORAL DOSAGE FORM WITH IONICALLY CHARGEABLE HYDROGEL FOR DELIVERY OF ACTIVE AGENT AND PERMEATION ENHANCER ENTREGA INC. (US) 2025-05-08 WO claimed
US-20250127723-A1 PHARMACEUTICAL COMPOSITION COMPRISING LARGE PHYSIOLOGICALLY ACTIVE SUBSTANCE AND EXCIPIENT D&D PHARMATECH INC. (KR) 2025-04-24 US claimed
US-20250099412-A1 METHOD OF INHIBITING DEGRADING PROTEASE ACTIVITY IN AGING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2025-03-27 US claimed
WO-2025054715-A1 COVID-19 TRAP TECHNOLOGY PLATFORM UNIVERSITY OF MANITOBA (CA) 2025-03-20 WO claimed
EP-1874726-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2008-01-09 EP claimed
EP-1210063-A4 COMPOSITIONS AND METHODS FOR ENHANCED ABSORPTION OF HYDROPHILIC THERAPEUTIC AGENTS LIPOCINE INC (US) 2007-08-15 EP claimed
WO-2006108643-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2006-10-19 WO claimed
US-7045323-B2 Glutathione reductase for therapy and prophylaxis of aids ANSOVINI RAFFAELE 2006-05-16 US claimed
WO-2005023835-A2 MODULATORS OF TRANSMEMBRANE PROTEASE SERINE 6 IRM LLC (BM) 2005-03-17 WO claimed
US-20050054027-A1 Modulators of transmembrane protease serine 6 IRM LLC (BM) 2005-03-10 US claimed
US-20040223958-A1 Glutathione reductase for therapy and prophylaxis of AIDS ANSOVINI RAFFAELE (IT) 2004-11-11 US claimed
EP-1210063-A1 COMPOSITIONS AND METHODS FOR ENHANCED ABSORPTION OF HYDROPHILIC THERAPEUTIC AGENTS Lipocine, Inc. (US) 2002-06-05 EP claimed
US-6309663-B1 Triglyceride-free compositions and methods for enhanced absorption of hydrophilic therapeutic agents LIPOCINE INC. 2001-10-30 US claimed
WO-2001012155-A1 COMPOSITIONS AND METHODS FOR ENHANCED ABSORPTION OF HYDROPHILIC THERAPEUTIC AGENTS LIPOCINE, INC. (US) 2001-02-22 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250188022-A1 PROCESS FOR THE PREPARATION OF NAFAMOSTAT, CAMOSTAT AND THEIR DERIVATIVES TPMT, ADH1C, ADH1A F2 1213/4885ADRA1A 3293/4885PRSS1 1209/4885
US-20260139860-A1 PRODUCTS OF MANUFACTURE FOR THE TREATMENT, PREVENTION AND AMELIORATION OF MICROBIAL INFECTIONS ACE, MAVS, SARS1 F2 828/4885ADRA1A 2150/4885PRSS1 281/4885
US-20250127723-A1 PHARMACEUTICAL COMPOSITION COMPRISING LARGE PHYSIOLOGICALLY ACTIVE SUBSTANCE AND EXCIPIENT CYP7A1, CYP11B1, CYP11B2 F2 524/4885ADRA1A 408/4885PRSS1 791/4885
US-12458622-B2 Methods of treatment of coronavirus-induced inflammation conditions C3AR1, IL5, IL4 F2 265/4885ADRA1A 2098/4885PRSS1 236/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.