SCHEMBL8719876

SCHEMBL8719876

CCCCc1nc(Cl)c(C=O)n1Cc1ccc2nc(-c3ccccc3C(=O)OC)ccc2c1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 4/20 0.57
AGTR2 P50052 4/20 0.57
GP6 Q9HCN6 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8916330 0.91 AGTR1 (0.62) AGTR1AGTR2
SCHEMBL8913829 0.90 AGTR1 (0.61) AGTR1AGTR2
SCHEMBL8326292 0.90 AGTR1 (0.59) AGTR1AGTR2GP6
SCHEMBL8913822 0.89 AGTR1 (0.58) AGTR1AGTR2GP6
SCHEMBL359 0.88 GP6 (0.63) AGTR1AGTR2GP6
SCHEMBL8914300 0.88 AGTR2 (0.64) AGTR1AGTR2
SCHEMBL8792485 0.86 AGTR1 (0.64) AGTR1AGTR2GP6
SCHEMBL8913133 0.82 ALDH1A1 (0.50) AGTR1AGTR2
SCHEMBL9694822 0.80 AGTR1 (0.57) AGTR1AGTR2GP6
SCHEMBL8912755 0.80 GP6 (0.55) AGTR1AGTR2GP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-6016659-A None JP disclosed
EP-0693478-B1 Quinoline compounds GREEN CROSS CORP (JP) 1998-08-12 EP disclosed
US-5665881-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE, ANGIOTENSIN II ANTAGONIST THE GREEN CROSS CORPORATION (JP) 1997-09-09 US disclosed
EP-0693478-A1 Quinoline compounds THE GREEN CROSS CORPORATION (JP) 1996-01-24 EP disclosed
US-5478832-A Angiotensin II antagonists; cardiovascular disorders THE GREEN CROSS CORPORATION (JP) 1995-12-26 US disclosed
JP-H0616659-A QUINOLINE DERIVATIVE ASAHI GLASS CO LTD 1994-01-25 JP disclosed
EP-0569013-A1 Quinoline compounds as angiotensin II antagonists THE GREEN CROSS CORPORATION (JP) 1993-11-10 EP disclosed
JP-H00616659-A 0001-01-01 JP disclosed