SCHEMBL8722148

SCHEMBL8722148

O=[N+]([O-])c1cccc(-c2cc(Br)c(-n3ccnc3)s2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.41
CHRNA5 P30532 1/20 0.41
CHRNA4 P43681 1/20 0.41
PKM P14618 2/20 0.40
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
RAB9A P51151 5/20 0.40
MAPT P10636 4/20 0.40
NPC1 O15118 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTPN1 P18031 1/20 0.39
PDE4B Q07343 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726099 0.87 PKM (0.41) PKMMGAMGAASIMGAM2
SCHEMBL8720881 0.83 MEN1 (0.47) MAPTCYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8720919 0.82 MAPT (0.46) PKMMGAMGAASIMGAM2
SCHEMBL8722162 0.81 PKM (0.36) CHRNB2CHRNA5CHRNA4PKMMGAM
SCHEMBL8722302 0.80 MGAM (0.42) PKMMGAMGAASIMGAM2
SCHEMBL8721485 0.75 NOTUM (0.47) CYP1A2CYP3A4SMN1; SMN2ALDH1A1LMNA
SCHEMBL8724367 0.75 LMNA (0.48) PKMMGAMGAASIMGAM2
SCHEMBL2627217 0.72 IDO1 (0.59) MAPTCYP3A4ALDH1A1LMNAMEN1
SCHEMBL31463543 0.70 GRIK1 (0.46) GAAMAPTKMT2APDE5A
SCHEMBL8726103 0.68 MEN1 (0.49) GAAMAPTCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998000430-A1 IMIDAZOL DERIVATIVES USEFUL AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-01-08 WO disclosed