SCHEMBL8734217

SCHEMBL8734217

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)C(F)(F)C(=O)N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.46
CTSS P25774 2/20 0.46
CTSB P07858 1/20 0.46
CTSK P43235 1/20 0.46
TACR2 P21452 5/20 0.45
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
HTRA1 Q92743 2/20 0.44
YAP1 P46937 3/20 0.43
MME P08473 1/20 0.43
ACE P12821 1/20 0.43
CPA1 P15085 1/20 0.43
ACE2 Q9BYF1 1/20 0.43
CMA1 P23946 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8735984 0.86 CTSD (0.49) CTSSCTSBCTSKTACR2ITGB3
SCHEMBL8041651 0.82 MME (0.47) CTSSCTSKITGB3ITGA2BMME
SCHEMBL8736216 0.82 CTSD (0.53) CTSSCTSKITGB3ITGA2BHTRA1
SCHEMBL8945318 0.82 CTSD (0.46) CTSSCTSKITGB3ITGA2BHTRA1
SCHEMBL8945610 0.81 MME (0.45) CTSSCTSKITGB3ITGA2BMME
SCHEMBL7422223 0.80 ITGB3 (0.45) CTSSCTSKITGB3ITGA2BMME
SCHEMBL8892233 0.80 ITGB3 (0.50) CTSSCTSBCTSKITGB3ITGA2B
SCHEMBL7933938 0.80 CTSD (0.47) RENCTSSCTSBCTSKITGB3
SCHEMBL8945566 0.80 CTSD (0.47) RENCTSSCTSBCTSKITGB3
SCHEMBL8492505 0.80 MME (0.64) ITGB3ITGA2BMMEACECPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716973-A ADMINISTERING DIFLUORO STATONE ANALOGS MERRELL PHARMACEUTICALS INC. (US) 1998-02-10 US disclosed
US-5559140-A VIRICIDES MERRELL PHARMACEUTICALS INC. (US) 1996-09-24 US disclosed
EP-0565631-B1 ANTI-VIRAL COMPOUNDS MERRELL PHARMA INC (US) 1996-09-18 EP disclosed
EP-0565631-A1 ANTI-VIRAL COMPOUNDS. MERRELL DOW PHARMA (US) 1993-10-20 EP disclosed
WO-1992012123-A1 ANTI-VIRAL COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-07-23 WO disclosed