SCHEMBL8744837

SCHEMBL8744837

COC(=O)[C@@H](NC(=O)Cc1c(C)cc(C)cc1C)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.49
TAS1R1 Q7RTX1 2/20 0.49
ALDH1A1 P00352 6/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
THRB P10828 1/20 0.42
HTT P42858 1/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PSMB5 P28074 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594891 1.00 TAS1R3 (0.49) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2
SCHEMBL6993048 0.91 TAS1R3 (0.44) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2
SCHEMBL7950138 0.91 TAS1R3 (0.44) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2
SCHEMBL7964617 0.90 TAS1R3 (0.48) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2
SCHEMBL6990364 0.90 TAS1R3 (0.48) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2
SCHEMBL8744786 0.90 ALDH1A1 (0.42) TAS1R3TAS1R1ALDH1A1SMN1; SMN2THRB
SCHEMBL9595171 0.90 ALDH1A1 (0.42) TAS1R3TAS1R1ALDH1A1SMN1; SMN2THRB
SCHEMBL8744706 0.85 THRA (0.45) NPSR1THRBMEN1KMT2APSMB5
SCHEMBL8744704 0.85 THRA (0.45) NPSR1THRBMEN1KMT2APSMB5
SCHEMBL27407409 0.82 TAS1R3 (0.44) TAS1R3TAS1R1ALDH1A1NPSR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed