Water

Water

SCHEMBL87641

C(=C1CCO1)c1ccccc1.O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
CYP1A2 P05177 2/20 0.43
F3 P13726 1/20 0.41
KDM4E B2RXH2 4/20 0.41
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.38
MAOB P27338 2/20 0.37
HPGD P15428 4/20 0.36
LMNA P02545 1/20 0.36
DYRK1A Q13627 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
GRM5 P41594 1/20 0.35
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3056491 0.98 ALDH1A1 (0.59) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL28305385 0.87 ALDH1A1 (0.48) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL28575414 0.81 ALDH1A1 (0.56) ALDH1A1CYP1A2F3KDM4EHTT
Methylsulfanylmethane SCHEMBL28306521 0.81 ALDH1A1 (0.43) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL28575415 0.81 ALDH1A1 (0.56) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL3069464 0.78 ALDH1A1 (0.47) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL9987943 0.77 PPARG (0.44) ALDH1A1CYP1A2F3KDM4EKMT2A
SCHEMBL14917485 0.76 ALDH1A1 (0.43) ALDH1A1CYP1A2F3HTTKMT2A
SCHEMBL3526528 0.72 ALDH1A1 (1.00) ALDH1A1CYP1A2F3KDM4EHTT
SCHEMBL981190 0.72 ALDH1A1 (1.00) ALDH1A1CYP1A2F3KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 151 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9388300-B2 High structure carbon blacks CABOT CORPORATION (US) 2016-07-12 US claimed
US-12018162-B2 Acrylic polymers for inkjet ink applications CABOT CORPORATION (US) 2024-06-25 US disclosed
EP-3294813-B1 AMPHOTERIC POLYMERS AND USE IN INKJET INK COMPOSITIONS CABOT CORP (US) 2024-06-12 EP disclosed
EP-4248010-A1 DIGITAL TEXTILE PRINTING INKS HAVING ZERO VOLATILE ORGANIC COMPOUND SOLVENTS THEREIN International Imaging Materials Inc. (US) 2023-09-27 EP disclosed
WO-2022108648-A1 DIGITAL TEXTILE PRINTING INKS HAVING ZERO VOLATILE ORGANIC COMPOUND SOLVENTS THEREIN INTERNATIONAL IMAGING MATERIALS, INC. (US) 2022-05-27 WO disclosed
US-20220154019-A1 DIGITAL TEXTILE PRINTING INKS HAVING ZERO VOLATILE ORGANIC COMPOUND SOLVENTS THEREIN INTERNATIONAL IMAGING MATERIALS, INC. (US) 2022-05-19 US disclosed
US-20220153047-A1 DIGITAL TEXTILE PRINTING INKS HAVING ZERO VOLATILE ORGANIC COMPOUND SOLVENTS THEREIN INTERNATIONAL IMAGING MATERIALS, INC. (US) 2022-05-19 US disclosed
US-20220010152-A1 POLYMERS FOR INKJET INK COMPOSITIONS CABOT CORP (US) 2022-01-13 US disclosed
US-20210395548-A1 ACRYLIC POLYMERS FOR INKJET INK APPLICATIONS CABOT CORPORATION 2021-12-23 US disclosed
US-20210324214-A1 DURABLE OUTDOOR INKJET INKS INTERNATIONAL IMAGING MATERIALS, INC. (US) 2021-10-21 US disclosed
EP-0943666-B1 Ink, ink set, ink cartridge, recording unit, image recording apparatus and image recording method CANON KK (JP) 2006-09-27 EP disclosed
US-20060211791-A1 Inkjet inks comprising modified pigments having attached polymeric groups CABOT CORPORATION 2006-09-21 US disclosed
WO-2006086660-A1 INKJET INKS COMPRISING MODIFIED PIGMENTS HAVING ATTACHED POLYMERIC GROUPS CABOT CORPORATION (US) 2006-08-17 WO disclosed
EP-1354921-A2 Process for alleviating bleeding between a black image and a color image during ink jet printingd CANON KABUSHIKI KAISHA (JP) 2003-10-22 EP disclosed
US-6332919-B2 SELF DISPERSABLE CARBON BLACK THAT HAS HYDROPHILIC GROUPS DIRECTLY OR VIA OTHER ATOMIC GROUPS ATTACHED TO ITS SURFACE AND VARIOUS ORGANIC OR INORGANIC SALTS; COLORFASTNESS CANON KABUSHIKI KAISHA (JP) 2001-12-25 US disclosed
US-20010020431-A1 Ink, Ink set, ink cartridge, recording unit, image recording apparatus and image recording method OSUMI KOICHI (JP) 2001-09-13 US disclosed
US-6280513-B1 OPTICAL RECORDING MEDIA; MIXTURE OF CARBON BLACK AND SALT CANON KABUSHIKI KAISHA (JP) 2001-08-28 US disclosed
EP-0943666-A2 Ink, ink set, ink cartridge, recording unit, image recording apparatus and image recording method CANON KABUSHIKI KAISHA (JP) 1999-09-22 EP disclosed
US-5843620-A Image-forming material KONICA CORPORATION (JP) 1998-12-01 US disclosed
US-5736286-A SWELLING TO WEAKEN ADHESION BETWEEN THE DEPOSITED IMAGES AND RECORDING MATERIAL RICOH COMPANY, LTD. (JP) 1998-04-07 US disclosed