SCHEMBL8767144

SCHEMBL8767144

CCN(CC)C(=O)c1ccc(S(=O)(=O)NC(=O)c2cnc(OC(=O)NCC(=O)O)c(OCC(C)C)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SCN9A Q15858 5/20 0.37
SCN5A Q14524 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.35
NAMPT P43490 1/20 0.35
EGFR P00533 2/20 0.35
LIMK1 P53667 1/20 0.35
LIMK2 P53671 1/20 0.35
PTGS2 P35354 1/20 0.34
P4HTM Q9NXG6 1/20 0.34
RXRA P19793 1/20 0.34
PPARG P37231 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099449 0.91 LMNA (0.37) LMNAHPGDHTTSMN1; SMN2SCN9A
SCHEMBL8767162 0.90 LMNA (0.40) LMNAHPGDHTTSMN1; SMN2SCN9A
SCHEMBL8917435 0.88 LMNA (0.38) LMNAHPGDHTTSMN1; SMN2L3MBTL1
SCHEMBL8768423 0.87 LMNA (0.41) LMNAHPGDHTTSMN1; SMN2L3MBTL1
SCHEMBL8768258 0.84 CA1 (0.39) SCN9AEGFRLIMK1LIMK2PTGS2
SCHEMBL8767453 0.83 LMNA (0.42) LMNAHPGDHTTSMN1; SMN2L3MBTL1
SCHEMBL8768350 0.83 MAPT (0.44) LMNAHTTSMN1; SMN2PTGS2
SCHEMBL8097664 0.83 ABL1 (0.37) LMNAHPGDHTTSMN1; SMN2SCN9A
SCHEMBL8096944 0.81 SMN1; SMN2 (0.39) LMNAHPGDHTTSMN1; SMN2SCN9A
SCHEMBL8875047 0.79 SMN1; SMN2 (0.36) LMNAHPGDHTTSMN1; SMN2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673931-B1 Sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AG (DE) 1997-08-13 EP disclosed
EP-0673931-A1 Sulfonamidocarbonyl-pyridine-2-carboxamides and their pyridine-N-oxides, process for their preparation and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-09-27 EP disclosed